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Apitolisib, MedChemExpress

Product Code. 16496126
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Product Code. 16496126 Supplier Medchem Express Supplier No. HY13246

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Description

MedChemExpress Apitolisib (GDC-0980; GNE 390; RG 7422) is a selective, potent, orally bioavailable Class I PI3 kinase and mTOR kinase (TORC1/2) inhibitor with IC50s of 5 nM/27 nM/7 nM/14 nM for PI3Kα/PI3Kβ/PI3Kδ/PI3Kγ, and with a Ki of 17 nM for mTOR.

Apitolisib (GDC-0980

Specifications

Chemical Name or Material Apitolisib
Physical Form Solid
CAS 1032754-93-0
Color Yellow
Quantity 100 mg
Purity Grade Notes Research
Molecular Formula C23H30N8O3S
For Use With (Application) Cancer-Kinase/protease
Synonym GDC-0980 GNE 390 RG 7422
Solubility Information DMSO : 14.29 mg/mL (28.66 mM; Need ultrasonic)
SMILES C[C@@H](C(N1CCN(CC1)CC2=C(C3=NC(C4=CN=C(N=C4)N)=NC(N5CCOCC5)=C3S2)C)=O)O
Molecular Weight (g/mol) 498.6
Formula Weight 498.6
Percent Purity 97.88%
Grade Research
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Research purposes only

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