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KDM5A-IN-1, MedChemExpress

Product Code. 16482738
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Product Code. 16482738

Brand: Medchem Express HY100014

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Description

MedChemExpress KDM5A-IN-1 is a potent, orally bioavailable pan-histone lysine demethylases 5 (KDM5) inhibitor with IC50s of 45 nM, 56 nM and 55 nM for KDM5A, KDM5B and KDM5C, respectively, and with an EC50 value of 960 nM for PC9 H3K4Me3. KDM5A-IN-1 is significantly less potent against other KDM5B enzymes (1A, 2B, 3B, 4C, 6A, 7B).

KDM5A-IN-1 is a potent, orally bioavailable pan-histone lysine demethylases 5 (KDM5) inhibitor with IC50s of 45 nM, 56 nM and 55 nM for KDM5A, KDM5B and KDM5C, respectively, and with an EC50 value of 960 nM for PC9 H3K4Me3. KDM5A-IN-1 is significantly less potent against other KDM5B enzymes (1A, 2B, 3B, 4C, 6A, 7B).

Specifications

Chemical Name or Material KDM5A-IN-1
Physical Form Powder
CAS 1905481-36-8
Color Off-White
Quantity 10 mg
Purity Grade Notes Research
Molecular Formula C15H22N4O2
For Use With (Application) Cancer-programmed cell death
Solubility Information DMSO : ≥ 50 mg/mL (172.20 mM)
SMILES O=C(C1CC1)N[C@@H]2CCN(C(C3=CC(C(C)C)=NN3)=O)C2
Molecular Weight (g/mol) 290.36
Formula Weight 290.36
Percent Purity 95.71%
Grade Research
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Research purposes only

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