missing translation for 'onlineSavingsMsg'
Learn More
  1. Home
  2. Products
  3. Cell Culture Media, Supplements, and Reagents
  4. Cell Culture Reagents, Antibiotics and Supplements
  5. Antibiotics
  6. LY2183240, MedChemExpress

LY2183240, MedChemExpress

Product Code. 16464218
Encompass_Preferred
Change view
Click to view available options
Quantity:
10 mg
50 mg
Unit Size:
10mg
50mg
2 product options available for selection
Product selection table with 2 available options. Use arrow keys to navigate and Enter or Space to select.
Product Code. Quantity unitSize
16464218 10 mg 10mg
16460557 50 mg 50mg
Use arrow keys to navigate between rows. Press Enter or Space to select a product option. 2 options available.
2 options
This item is not returnable. View return policy
Product Code. 16464218 Supplier Medchem Express Supplier No. HY10865

Please to purchase this item. Need a web account? Register with us today!

This item is not returnable. View return policy

Description

MedChemExpress LY2183240 is a highly potent blocker of anandamide uptake (IC50= 270 pM; Ki=540 nM).

LY2183240 is a potent, covalent inhibitor of the endocannabinoid-degrading enzyme fatty acid amide hydrolase (FAAH) with an IC50 of 12.4 nM. LY2183240 inactivates FAAH by carbamylation of the enzyme's serine nucleophile. LY2183240 also inhibits several other brain serine hydrolases with IC50s of 5.3, 0.09, 8.2 nM for MAG lipase, bh6 and KIAA1363, respectively .

Specifications

Chemical Name or Material LY2183240
Physical Form Solid
CAS 874902-19-9
Color Light Yellow
Quantity 10 mg
Purity Grade Notes Research
Molecular Formula C17H17N5O
For Use With (Application) Neuroscience-Neuromodulation
Solubility Information DMSO : 50 mg/mL (162.68 mM; Need ultrasonic)
SMILES O=C(N(C)C)N1N=NN=C1CC(C=C2)=CC=C2C3=CC=CC=C3
Molecular Weight (g/mol) 307.35
Formula Weight 307.35
Percent Purity 98.01%
Grade Research
Show More Show Less

Research purposes only

Product Title
Select an issue

By clicking Submit, you acknowledge that you may be contacted by Fisher Scientific in regards to the feedback you have provided in this form. We will not share your information for any other purposes. All contact information provided shall also be maintained in accordance with our Privacy Policy.